Aromasin (Exemestane) to improve body proportions

by adnorthfloridaho
March 25, 2022
1406

Bodybuilders are very inventive in synergistic drug combinations. The symbiosis of anabolic steroids, growth hormone and insulin created the first athletes with mountains of muscle. So, many people combine exemestane with selective estrogen receptor modifiers (SERMs), steroids, and GH, and thus achieve good results. On the forums, it comes to anecdotal confessions about the results of blood tests and the achievements of this or that athlete against the background of these results.

Aromasin (Exemestane) is an aromatase inhibitor that reduces the production of estrogen in the body. This drug is approved in the US for the treatment of breast cancer.

In bodybuilding, Aromasin (Exemestane) is used on a steroid course to reduce the aromatous effect (converting testosterone to estrogen) when taking anabolic hormonal drugs.

Effects of Aromasin (Exemestane)

Prevention of gynecomastia
Decreased estrogen production (by 97%)4
Increasing anabolic hormone levels
Improving the relief of muscles
Prevention of hypertension

Dosages and course of taking Aromasin (Exemestane)

For prevention (in bodybuilding): 12.5 mg every other day.
For the treatment of gynecomastia: 25 mg every day until the symptoms disappear (then 12.5 mg every other day).

Taking a course of steroids:

When using steroids with a short half-life (testosterone propionate, methandrostenolone): after 10 days of the course, take an analysis for estradiol and take 12.5 mg of Aromasin (Exemestane) every other day. Then, after 10 days, once again take tests for estradiol and adjust the dosage of Aromasin (Exemestane) according to their results.
When using steroids with long esters (enanthate, sustanon, cypionate): after 3-4 weeks of the course, take tests for estradiol and take 12.5 mg of Aromasin (Exemestane) every other day. Then, after 10 days, once again take tests for estradiol and adjust the dosage of Aromasin (Exemestane) according to their results.

Like other aromatase inhibitors, the dosage of Aromasin can be adjusted according to subjective feelings. If depression, a drop in libido and erectile dysfunction are observed while taking Aromasin (Exemestane), the dosage should be reduced.

Read also about Aromasin dosage

Side effects of Aromasin (Exemestane)

Exceeding dosages and abuse of aromatase inhibitors leads to excessive suppression of estrogen production and the following effects:

Nausea
Increased risk of fractures (by 60%)
Joint pain
Formation of arterial and venous thrombi
Dryness of the mucous membranes of the urogenital zone

Important! When using any pharmacological agents, it is recommended to consult a doctor.

When taking a course of steroids, you must strictly adhere to the rules listed below:

If an athlete uses steroids with a short half-life, ten days after the start of the course, tests must be performed to check the concentration of estradiol in the body. Next, you need to take Exemestane Grindeks at a dosage of 12.5 milligrams. Periodicity – day after day. After another ten days, an identical analysis is required again. Depending on the results obtained, it is necessary to either adjust the dosage, or continue the course according to an identical scheme;

Read also about aromasin dosage bodybuilding

As part of taking steroids, the composition of which includes long esters, it is necessary to pass an analysis to check the amount of estradiol a month after the start of the course. The dosage of Examestan is identical to the first rule. Ten days later, the athlete retakes the same analysis, according to the results of which the dosage is adjusted, or the dosage remains identical.

As in the case of other types of aromatase inhibitors, adjustment of the dosage of Examestan is allowed taking into account subjective sensations. The instruction for use attached to the drug Exemestane states the need to reduce the dose if a depressive state is observed, an erection is disturbed with a drop in libido.

“Aromatase inhibitors may well be an attractive alternative to replace the traditional hormone testosterone in the elderly, as these inhibitors can be taken orally once a day and can promote testosterone production in the body. In addition, abuse of aromatase inhibitors is unlikely as testosterone will not be stimulated to very high supraphysiological levels.

Read also about Aromasin users

One small experiment demonstrated that anastrozole at 1 mg per day for 12 weeks resulted in a doubling of low bioavailable testosterone levels in a group of older adults.

Another recent experiment also showed a moderate but significant effect of aromatase inhibition on estradiol and testosterone in the elderly. Atamestane 100mg once daily resulted in a 40% increase in total testosterone over a 36 week course. However, no positive impact on strength, muscle and other indicators was found.

A similar increase in testosterone levels, with no effect on body composition and strength performance, was documented in a study in which elderly men with borderline low serum testosterone levels were treated with anastrozole for 1 year.

“Blockade of estrogen action is a form of indirect activation of androgens that can stimulate a sustained but modest increase in endogenous luteinizing hormone (LH) secretion and makes it acceptable to maintain a modest increase in blood testosterone concentrations.

Therefore, it is likely that more effective estrogen blockade in men will produce a significant and sustained increase in blood testosterone levels, perhaps sufficient to achieve myotropic and stimulatory effects in men taking such drugs. Therefore, despite the lack of direct ergogenic studies regarding estrogen blockers in men, the available observations suggest that the use of estrogen blockers in relation to men is inappropriate.

Exemestane is a steroidal aromatase inhibitor sold under the brand name Aromasin. Unlike anastrozole and letrozole, which reversibly block aromatase, exemestane completely deactivates this enzyme by binding to its molecules. Inhibition of aromatase by Aromasin leads to a significant decrease in the level of estradiol in the blood, which makes the drug effective in the treatment of breast cancer. Due to its effectiveness, exemestane has also found its way into bodybuilding.

Aromasin is available in 25 mg tablets. The dosage of Aromasin on a course of steroids is usually 12.5 mg every other day, 12.5 mg per day, or, very rarely, 25 mg per day. It all depends on the individual reaction of the body. Competitive athletes take 25 mg/day in the last 7-14 days before competition to stiffen the muscles.

Bodybuilders are very inventive in synergistic drug combinations. The symbiosis of anabolic steroids, growth hormone and insulin created the first athletes with mountains of muscle. So, many people combine exemestane with selective estrogen receptor modifiers (SERMs), steroids, and GH, and thus achieve good results. On the forums, it comes to anecdotal confessions about the results…